SCHEMBL4680644

SCHEMBL4680644

[CH]1CNC(C2=NCCN2)=N1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 14/20 0.45
LMNA P02545 1/20 0.41
RECQL P46063 1/20 0.41
TOP2A P11388 1/20 0.40
TOP2B Q02880 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3742115 0.78 NISCH (0.56) NISCHLMNARECQLTOP2ATOP2B
SCHEMBL6992574 0.67 NISCH (0.72) NISCHLMNARECQLTOP2ATOP2B
SCHEMBL5476725 0.67 NISCH (0.79) NISCHLMNARECQLTOP2ATOP2B
SCHEMBL9375560 0.65 NISCH (0.61) NISCH
SCHEMBL16863098 0.65 NISCH (0.76) NISCH
SCHEMBL202587 0.64 NISCH (0.48) NISCHLMNARECQLTOP2ATOP2B
SCHEMBL9579892 0.64 NISCH (0.81) NISCH
SCHEMBL28428254 0.63 NISCH (0.60) NISCHTOP2ATOP2B
SCHEMBL105024 0.62 NISCH (1.00) NISCHLMNARECQLTOP2ATOP2B
SCHEMBL13167154 0.62 NISCH (0.47) NISCHLMNARECQLTOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142872-B1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO (JP) 2008-10-15 EP disclosed
EP-1142872-A1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO., LTD. (JP) 2001-10-10 EP disclosed