SCHEMBL4681372

SCHEMBL4681372

COCCOc1cc(=O)c(O)c2n1CCN(Cc1ccc(F)c(Cl)c1)C2=O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 3/20 0.38
P2RX7 Q99572 2/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
ERCC1 P07992 1/20 0.35
ERCC4 Q92889 1/20 0.35
TNIK Q9UKE5 1/20 0.34
HTR2A P28223 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
DRD4 P21917 1/20 0.34
PDE4A P27815 1/20 0.34
KCNH2 Q12809 1/20 0.33
CLPP Q16740 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687652 0.91 MAOB (0.39) GRM2KDM4EALDH1A1HPGDHTT
SCHEMBL4684887 0.80 MAOB (0.42) KDM4EALDH1A1HPGDHTTERCC1
SCHEMBL4683024 0.79 NAMPT (0.39) GRM2P2RX7KDM4EALDH1A1HPGD
SCHEMBL5522450 0.78 ERCC1 (0.39) P2RX7ERCC1ERCC4KCNH2CLPP
SCHEMBL3907766 0.78 ERCC1 (0.44) GRM2P2RX7ERCC1ERCC4TNIK
SCHEMBL5529791 0.77 ERCC1 (0.36) GRM2P2RX7KDM4EALDH1A1HPGD
SCHEMBL4682670 0.76 P2RX7 (0.43) GRM2P2RX7KDM4EALDH1A1KCNH2
SCHEMBL2895650 0.75 MAOB (0.38) GRM2P2RX7KDM4EALDH1A1HPGD
SCHEMBL4318863 0.74 MAOB (0.41) KDM4EALDH1A1HPGDHTTERCC1
SCHEMBL4684845 0.74 KCNH2 (0.40) GRM2P2RX7ALDH1A1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973906-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE Virochem Pharma Inc. (CA) 2008-10-01 EP claimed
WO-2006066414-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2006-06-29 WO claimed
EP-1973906-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE Virochem Pharma Inc. (CA) 2008-10-01 EP disclosed
WO-2006066414-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2006-06-29 WO disclosed