SCHEMBL4684845

SCHEMBL4684845

O=C1c2c(O)c(=O)cc(OCC(F)(F)F)n2CCN1Cc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.40
GRM2 Q14416 2/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
AKR1B1 P15121 1/20 0.38
LMNA P02545 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
HTT P42858 3/20 0.38
ALDH1A1 P00352 2/20 0.38
RAB9A P51151 1/20 0.38
CYP2D6 P10635 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
POLB P06746 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4681422 0.84 CYP2D6 (0.41) KCNH2GRM2MEN1KMT2AAKR1B1
SCHEMBL4682779 0.82 GRM2 (0.44) KCNH2GRM2MEN1KMT2AAKR1B1
SCHEMBL4682670 0.80 P2RX7 (0.43) KCNH2GRM2ALDH1A1RAB9AP2RX7
SCHEMBL4161790 0.76 MEN1 (0.44) KCNH2GRM2MEN1KMT2AAKR1B1
SCHEMBL2891898 0.75 KCNH2 (0.42) KCNH2GRM2MEN1KMT2AAKR1B1
SCHEMBL3905975 0.75 KCNH2 (0.46) KCNH2GRM2MEN1KMT2AAKR1B1
SCHEMBL4681372 0.74 GRM2 (0.38) KCNH2GRM2MEN1KMT2AHTT
SCHEMBL14129855 0.73 KCNH2 (0.39) KCNH2GRM2MEN1KMT2AAKR1B1
SCHEMBL4687652 0.72 MAOB (0.39) KCNH2GRM2SMN1; SMN2L3MBTL1HTT
Hydrochloric Acid SCHEMBL4324964 0.72 KCNH2 (0.38) KCNH2GRM2MEN1KMT2AAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973906-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE Virochem Pharma Inc. (CA) 2008-10-01 EP disclosed
WO-2006066414-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2006-06-29 WO disclosed