SCHEMBL4684092

SCHEMBL4684092

CCc1cc([N+](=O)[O-])ccc1C(=O)N1CCCC(OCCO)c2cc(F)ccc21

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.36
ALDH1A1 P00352 8/20 0.36
MAPT P10636 6/20 0.36
LMNA P02545 3/20 0.36
GAA P10253 1/20 0.36
HTT P42858 3/20 0.35
NPC1 O15118 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
NPY2R P49146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7342308 0.91 MAPT (0.39) WDR5ALDH1A1MAPTLMNAHTT
SCHEMBL4681210 0.86 MAPT (0.38) WDR5ALDH1A1MAPTLMNAHTT
Iodide SCHEMBL4686142 0.80 AVPR2 (0.40) WDR5ALDH1A1MAPTLMNAHTT
SCHEMBL4686569 0.80 MEN1 (0.41) ALDH1A1MAPTLMNAHTTNPC1
SCHEMBL4685743 0.80 RAB9A (0.37) WDR5ALDH1A1MAPTLMNAHTT
SCHEMBL7335351 0.79 ALDH1A1 (0.37) ALDH1A1MAPTLMNAGAAMEN1
SCHEMBL4687267 0.79 AVPR2 (0.43) ALDH1A1MAPTLMNAHTTNPC1
SCHEMBL4682375 0.77 ALDH1A1 (0.38) ALDH1A1MAPTLMNAHTTMEN1
SCHEMBL7333794 0.77 ALDH1A1 (0.41) WDR5ALDH1A1MAPTLMNAGAA
SCHEMBL5474822 0.77 MAPT (0.39) WDR5ALDH1A1MAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed