SCHEMBL4684237

SCHEMBL4684237

Cc1c(F)cc(C(=O)Nc2ccon2)cc1-c1ccc(C(N)=O)c(CC(C)(C)C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.39
KDM4E B2RXH2 3/20 0.39
GAA P10253 1/20 0.39
MAPK14 Q16539 7/20 0.38
SYK P43405 1/20 0.38
CYP2C9 P11712 4/20 0.38
BUB1 O43683 1/20 0.38
PRKACG P22612 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
MAPK11 Q15759 1/20 0.38
ACSL5 Q9ULC5 1/20 0.38
STK24 Q9Y6E0 1/20 0.38
LCK P06239 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 2/20 0.35
ALDH1A1 P00352 4/20 0.35
HPGD P15428 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HTT P42858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680753 0.78 MAPK14 (0.46) SMN1; SMN2KDM4EGAAMAPK14CYP2C9
SCHEMBL4681674 0.76 MAPK14 (0.66) SMN1; SMN2KDM4EGAAMAPK14CYP2C9
SCHEMBL14077653 0.73 SMN1; SMN2 (0.56) SMN1; SMN2KDM4EGAAMAPK14CYP2C9
SCHEMBL4740641 0.69 SMN1; SMN2 (0.54) SMN1; SMN2KDM4EGAAMAPK14CYP2C9
SCHEMBL4684166 0.69 SMN1; SMN2 (0.53) SMN1; SMN2KDM4EGAAMAPK14CYP2C9
SCHEMBL14077643 0.66 SMN1; SMN2 (0.47) SMN1; SMN2KDM4EGAAMAPK14CYP2C9
SCHEMBL14269565 0.66 ADORA2A (0.53) SMN1; SMN2MAPK14CYP2C9BUB1PRKACG
SCHEMBL3890906 0.64 SMN1; SMN2 (0.62) SMN1; SMN2KDM4EGAAMAPK14TSHR
SCHEMBL3637436 0.64 MAPK14 (0.82) SMN1; SMN2GAAMAPK14CYP2C9MAPKAPK2
SCHEMBL380138 0.62 MAPK14 (0.53) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891061-A1 N-(2, 2-DIMETHYLPROPYL) -6- (3-FLUORO-5- ( (3-ISOXAZOLYLAMINO) CARBONYL) -2-METHYLPHENY L) -3-PYRIDINECARBOXAMIDE SmithKline Beecham Corporation (US) 2008-02-27 EP disclosed
WO-2006134382-A1 N-(2, 2-DIMETHYLPROPYL) -6- (3-FLUORO-5- ( (3-ISOXAZOLYLAMINO) CARBONYL) -2-METHYLPHENY L) -3-PYRIDINECARBOXAMIDE SMITHKLINE BEECHAM CORPORATION (US) 2006-12-21 WO disclosed