SCHEMBL4686769

SCHEMBL4686769

CC(C)(C)COC(=O)NC(Cc1ccc2c(c1)NC(=O)[C@H](CCC(=O)OCc1ccccc1)O2)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.40
CTSK P43235 4/20 0.40
KLK7 P49862 1/20 0.38
KLK5 Q9Y337 1/20 0.38
IDO1 P14902 3/20 0.38
TDO2 P48775 1/20 0.38
CCKAR P32238 1/20 0.38
CCKBR P32239 1/20 0.38
EPHX2 P34913 1/20 0.38
CTSS P25774 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854525 0.93 IDO1 (0.43) CTSLCTSKIDO1TDO2CTSS
SCHEMBL4854521 0.93 IDO1 (0.43) CTSLCTSKIDO1TDO2CTSS
SCHEMBL4854530 0.93 IDO1 (0.43) CTSLCTSKIDO1TDO2CTSS
SCHEMBL4685497 0.90 USP2 (0.37) KLK5IDO1CCKARCCKBREPHX2
SCHEMBL7166021 0.89 ACE (0.47) CTSLCTSKKLK7KLK5IDO1
SCHEMBL7363235 0.89 KLK5 (0.42) CTSLCTSKKLK7KLK5IDO1
SCHEMBL4853017 0.83 ITGB3 (0.43) IDO1TDO2
SCHEMBL4852776 0.83 ITGB3 (0.43) IDO1TDO2
SCHEMBL4680620 0.83 ITGB3 (0.43) IDO1TDO2
SCHEMBL7169155 0.82 ITGB3 (0.46) CTSLCTSKIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594853-B1 METHOD FOR THE PRODUCTION OF BICYCLIC AROMATIC AMINO ACIDS AND INTERMEDIATE PRODUCTS THEREOF MERCK PATENT GMBH (DE) 2008-07-09 EP disclosed