SCHEMBL4688602

SCHEMBL4688602

Cc1cccc(C2=CCNCC2)c1C#N

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.46
HTR6 P50406 2/20 0.45
SIGMAR1 Q99720 2/20 0.44
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
DRD2 P14416 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GAA P10253 1/20 0.40
HTR2A P28223 1/20 0.40
HTT P42858 1/20 0.40
RAD52 P43351 1/20 0.40
KHK P50053 1/20 0.39
QDPR P09417 1/20 0.38
PIK3CD O00329 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4930633 1.00 HTR2C (0.46) HTR2CHTR6SIGMAR1KDM4EALDH1A1
SCHEMBL7566975 0.80 HTR2C (0.53) HTR2CHTR6SIGMAR1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL9530706 0.79 HTR2C (0.61) HTR2CHTR6SIGMAR1KDM4EALDH1A1
SCHEMBL1366798 0.79 HTR2C (0.61) HTR2CHTR6SIGMAR1KDM4EALDH1A1
SCHEMBL19297061 0.78 HTR2C (0.53) HTR2CHTR6SIGMAR1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL2176384 0.76 HTR2C (0.49) HTR2CHTR6SIGMAR1KHKQDPR
Hydrochloric Acid SCHEMBL29882704 0.75 HTR2C (0.56) HTR2CHTR6SIGMAR1KDM4EALDH1A1
SCHEMBL5317969 0.75 HTR2C (0.56) HTR2CHTR6SIGMAR1KDM4EALDH1A1
SCHEMBL5321408 0.75 HTR6 (0.59) HTR2CHTR6SIGMAR1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL2171943 0.75 HTR6 (0.59) HTR2CHTR6SIGMAR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828125-B1 ARYLPIPERAZINE DERIVATIVES AND THEIR USE AS LIGANGS SELECTIVE OF THE DOPAMINE D3 RECEPTOR BIOPROJET SOC CIV (FR) 2008-04-09 EP disclosed
EP-1828125-A1 ARYLPIPERAZINE DERIVATIVES AND THEIR USE AS LIGANGS SELECTIVE OF THE DOPAMINE D3 RECEPTOR BIOPROJET (FR) 2007-09-05 EP disclosed
WO-2006058993-A1 ARYLPIPERAZINE DERIVATIVES AND THEIR USE AS LIGANDS SELECTIVE OF THE DOPAMINE D3 RECEPTOR BIOPROJET (FR) 2006-06-08 WO disclosed