SCHEMBL4690039

SCHEMBL4690039

CC1(Cc2ccccc2)C(=O)N(c2cc(Cl)cc(Cl)c2)c2cccc(O)c21

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 12/20 0.70
ITGB2 P05107 11/20 0.70
ICAM1 P05362 11/20 0.70
ELANE P08246 2/20 0.50
PGR P06401 1/20 0.38
XIAP P98170 1/20 0.37
BIRC2 Q13490 1/20 0.37
TSHR P16473 1/20 0.37
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
THPO P40225 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690170 0.90 ITGAL (0.57) ITGALITGB2ICAM1
SCHEMBL4686803 0.90 ITGAL (0.57) ITGALITGB2ICAM1ELANE
SCHEMBL4689932 0.83 ITGAL (1.00) ITGALITGB2ICAM1ELANEPGR
SCHEMBL4686807 0.74 ITGAL (0.82) ITGALITGB2ICAM1ELANE
SCHEMBL13879533 0.69 ITGAL (0.76) ITGALITGB2ICAM1ELANETSHR
SCHEMBL4687618 0.68 ITGB2 (0.41) ITGALITGB2ICAM1ALDH1A1CYP1A2
SCHEMBL17716270 0.66 ELANE (0.87) ITGALITGB2ICAM1ELANEPGR
SCHEMBL13817154 0.64 ITGB2 (0.79) ITGALITGB2ICAM1
SCHEMBL17716269 0.63 ELANE (0.73) ITGALITGB2ICAM1ELANEPGR
SCHEMBL19184961 0.63 ELANE (0.73) ITGALITGB2ICAM1ELANEPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399155-B1 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMA (US) 2008-05-28 EP claimed
EP-1399155-A4 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMA (US) 2004-12-15 EP claimed
EP-1399155-A2 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-03-24 EP claimed
US-6414153-B1 TREATMENT OF INFLAMMATORY OR IMMUNE CELL-MEDIATED DISEASE OR CONDITION BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-07-02 US claimed
WO-2001006984-A2 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-02-01 WO claimed
EP-1399155-B1 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMA (US) 2008-05-28 EP disclosed
US-6414153-B1 TREATMENT OF INFLAMMATORY OR IMMUNE CELL-MEDIATED DISEASE OR CONDITION BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-07-02 US disclosed