Cyclopentane

Cyclopentane

SCHEMBL4690116

C1CCCC1.O=C(O)NC(CCN1CC2CN(Cc3ccc(Cl)c(Cl)c3)C[C@@H]2C1)c1ccccc1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.52
LIPG Q9Y5X9 1/20 0.47
FAAH O00519 1/20 0.47
SIGMAR1 Q99720 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
UTS2R Q9UKP6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclopentane SCHEMBL4695468 0.89 CCR5 (0.56) CCR5UTS2R
SCHEMBL4694382 0.80 SIGMAR1 (0.52) CCR5FAAHSIGMAR1MEN1KMT2A
SCHEMBL14435067 0.79 CCR5 (0.53) CCR5
Cyclopentane SCHEMBL4695436 0.78 CCR5 (0.62) CCR5
Cyclopentane SCHEMBL4695855 0.78 CCR5 (0.81) CCR5
Cyclopentane SCHEMBL4695395 0.78 CCR5 (0.68) CCR5
SCHEMBL13326659 0.78 CCR5 (0.75) CCR5
SCHEMBL13359857 0.78 CCR5 (0.75) CCR5
Cyclopentane SCHEMBL4695484 0.77 CCR5 (0.78) CCR5
Cyclopentane SCHEMBL4694741 0.76 CCR5 (0.60) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed