SCHEMBL4690601

SCHEMBL4690601

NC(=O)c1cc(-c2ccccc2)cc2c(C3=CCNCC3)c[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 16/20 0.56
CHUK O15111 3/20 0.56
CSF1R P07333 1/20 0.53
BTK Q06187 1/20 0.53
HTR2C P28335 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
DRD2 P14416 1/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48
SIGMAR1 Q99720 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688357 0.83 IKBKB (0.53) IKBKBCHUKCSF1RBTK
Hydrochloric Acid SCHEMBL1686965 0.82 HTR2C (0.43) IKBKBCHUKCSF1RBTKHTR2C
SCHEMBL10075358 0.82 HTR2C (0.43) IKBKBCHUKCSF1RBTKHTR2C
SCHEMBL4686046 0.81 IKBKB (0.62) IKBKBCHUKCSF1RBTK
SCHEMBL5306819 0.81 IKBKB (0.53) IKBKBCHUKHTR2CSIGMAR1
SCHEMBL3792407 0.77 HTR1A (0.56) IKBKBCHUKDRD2
SCHEMBL4688714 0.77 TDO2 (0.56) IKBKBCHUKBTK
SCHEMBL14030843 0.76 IKBKB (0.57) IKBKBCHUKCSF1RBTK
SCHEMBL7392593 0.74 JAK2 (0.69) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL4686501 0.74 IKBKB (0.54) IKBKBCHUKCSF1RBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1703905-B1 INDOLE DERIVATIVES AND USE THEREOF AS KINASE INHIBITORS IN PARTICULAR IKK2 INHIBITORS SMITHKLINE BEECHAM CORP (US) 2008-11-12 EP disclosed