SCHEMBL4690616

SCHEMBL4690616

COc1ccccc1-n1ncc(C(=O)N2CC3CN(CCC(=O)Nc4ccc(C)c(Cl)c4)CC3C2)c1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
HTT P42858 2/20 0.44
MAPT P10636 2/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MALT1 Q9UDY8 13/20 0.42
NR1H4 Q96RI1 1/20 0.42
TSHR P16473 2/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
SCN5A Q14524 1/20 0.41
SCN9A Q15858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690623 0.90 MAPT (0.42) MAPTLMNAMALT1NR1H4
SCHEMBL4691500 0.89 NR1H4 (0.54) ALDH1A1MAPTLMNAMALT1NR1H4
SCHEMBL4693420 0.87 MAPT (0.45) ALDH1A1MAPTLMNANR1H4TSHR
SCHEMBL4694220 0.86 NR1H4 (0.46) MAPTLMNAMALT1NR1H4GAA
SCHEMBL4695747 0.86 NR1H4 (0.47) MAPTLMNANR1H4KMT2A
SCHEMBL4692823 0.86 NR1H4 (0.47) MAPTLMNAL3MBTL1NR1H4GAA
SCHEMBL4691400 0.83 KMT2A (0.50) ALDH1A1HTTMAPTLMNATSHR
SCHEMBL4693690 0.81 HCRTR1 (0.51) ALDH1A1HTTMAPTLMNAGAA
SCHEMBL4693950 0.81 HCRTR1 (0.49) ALDH1A1HTTMAPTKMT2A
SCHEMBL4691680 0.80 POLB (0.52) MAPTNR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed