SCHEMBL4692823

SCHEMBL4692823

Cc1ccc(NC(=O)CCN2CC3CN(C(=O)c4cnn(-c5ccc(Cl)cc5)c4C(F)(F)F)CC3C2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.47
MAPT P10636 4/20 0.45
TP53 P04637 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 2/20 0.42
TRPC1 P48995 1/20 0.40
TRPC3 Q13507 1/20 0.40
STIM1 Q13586 1/20 0.40
ORAI1 Q96D31 1/20 0.40
STIM2 Q9P246 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
BLM P54132 1/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GPR6 P46095 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695747 0.95 NR1H4 (0.47) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4694220 0.95 NR1H4 (0.46) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4691500 0.94 NR1H4 (0.54) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4693420 0.93 MAPT (0.45) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4691333 0.89 MAPT (0.45) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4690616 0.86 ALDH1A1 (0.44) NR1H4MAPTGAAL3MBTL1LMNA
SCHEMBL4691661 0.85 MAPT (0.45) MAPTTP53SMN1; SMN2POLB
SCHEMBL4694966 0.84 NR1H4 (0.42) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4691680 0.83 POLB (0.52) NR1H4MAPTTP53SMN1; SMN2POLB
SCHEMBL4694232 0.83 PDK1 (0.42) NR1H4MAPTTP53SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed