SCHEMBL4690901

SCHEMBL4690901

COC(=O)C(N)(C(=O)Cc1ccccc1)P(=O)(OC)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.42
LAP3 P28838 1/20 0.39
KCNN4 O15554 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
PLAU P00749 1/20 0.38
ELANE P08246 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTPN1 P18031 2/20 0.37
CTRB1 P17538 1/20 0.37
GAA P10253 1/20 0.37
CES2 O00748 1/20 0.37
AKR1B1 P15121 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
NPC1 O15118 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL269403 0.82 PTPN1 (0.49) ALDH1A1RAB9ASMN1; SMN2PTPN1MEN1
SCHEMBL590493 0.82 PTPN1 (0.49) ALDH1A1RAB9ASMN1; SMN2PTPN1MEN1
SCHEMBL4687989 0.78 SRC (0.54) CES1KCNN4ALDH1A1KDM4ELMNA
SCHEMBL6120239 0.74 L3MBTL1 (0.34) KCNN4L3MBTL1
SCHEMBL11730655 0.73 CES1 (0.52) CES1KCNN4ALDH1A1KDM4ELMNA
SCHEMBL27815145 0.73 ALDH1A1 (0.45) LAP3ALDH1A1RAB9ASMN1; SMN2PTPN1
SCHEMBL5554985 0.70 PTPN1 (0.46) KCNN4ALDH1A1RAB9ASMN1; SMN2PTPN1
SCHEMBL16295744 0.69 SMN1; SMN2 (0.50) KCNN4ALDH1A1SMN1; SMN2PTPN1CTRB1
SCHEMBL12902954 0.69 CES1 (0.59) CES1ALDH1A1SMN1; SMN2CES2AKR1B1
SCHEMBL1874420 0.69 L3MBTL1 (0.31) ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581496-A4 2-SUBSTITUTED-3-PROPENAMIDE DERIVATIVES AND METHODS OF USING THE SAME GILEAD SCIENCES INC (US) 2008-04-23 EP disclosed
EP-1581496-A2 2-SUBSTITUTED-3-PROPENAMIDE DERIVATIVES AND METHODS OF USING THE SAME GILEAD SCIENCES, INC. (US) 2005-10-05 EP disclosed
WO-2004050613-A2 2-SUBSTITUTED-3-PROPENAMIDE DERIVATIVES AND METHODS OF USING THE SAME GILEAD SCIENCES, INC. (US) 2004-06-17 WO disclosed