SCHEMBL4691563

SCHEMBL4691563

Cc1ncnc(C)c1C(=O)N1CC2CN(CCNC(=O)c3cccc(F)c3)CC2C1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.58
CCL5 P13501 9/20 0.58
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694840 0.95 CCR5 (0.55) CCR5CCL5KCNH2
SCHEMBL4691570 0.86 CCR5 (0.59) CCR5CCL5KCNH2
SCHEMBL4972691 0.83 CCL5 (0.55) CCR5CCL5
SCHEMBL4695359 0.83 CCR5 (0.58) CCR5CCL5KCNH2
SCHEMBL14448125 0.80 CCR5 (0.72) CCR5CCL5KCNH2
SCHEMBL13326710 0.80 CCR5 (0.72) CCR5CCL5KCNH2
SCHEMBL4694606 0.79 CCR5 (0.49) CCR5CCL5
SCHEMBL4693572 0.79 CCR5 (0.70) CCR5CCL5KCNH2
SCHEMBL3286470 0.79 CCR5 (0.70) CCR5CCL5KCNH2
SCHEMBL3272374 0.79 CCR5 (0.70) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed