SCHEMBL4691995

SCHEMBL4691995

Cc1ccc(C(=O)NCCCN2CC3CN(C(=O)c4c(F)cccc4Cl)CC3C2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CCR5 P51681 2/20 0.43
SLC6A4 P31645 3/20 0.43
SLC6A2 P23975 1/20 0.43
RORC P51449 4/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
DRD2 P14416 2/20 0.42
DRD4 P21917 2/20 0.42
HTR1A P08908 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
DRD3 P35462 1/20 0.42
SMYD2 Q9NRG4 1/20 0.42
NPBWR1 P48145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691509 0.92 CCR5 (0.51) CCR5SLC6A4SLC6A2DRD2DRD4
SCHEMBL4695512 0.90 LMNA (0.41) SIGMAR1GAAALDH1A1SLC6A4SLC6A2
SCHEMBL4693309 0.89 LMNA (0.43) L3MBTL1GAAMAPTALDH1A1CCR5
SCHEMBL4694384 0.89 SLC6A4 (0.42) L3MBTL1SLC6A4SLC6A2HTR2AHTR2C
SCHEMBL4692216 0.89 SLC6A2 (0.43) GAASLC6A4SLC6A2DRD2DRD4
SCHEMBL4691999 0.86 MAPT (0.51) SIGMAR1GAAMAPTALDH1A1CCR5
SCHEMBL4691761 0.86 SLC6A2 (0.44) SLC6A4SLC6A2DRD2DRD4ADRA1A
SCHEMBL4695321 0.86 TSHR (0.43) MAPTALDH1A1
SCHEMBL4693332 0.85 SLC6A4 (0.45) SIGMAR1GAASLC6A4SLC6A2DRD2
SCHEMBL4691639 0.85 SMYD2 (0.48) SIGMAR1L3MBTL1ALDH1A1CCR5SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed