SCHEMBL4692691

SCHEMBL4692691

Cc1ccc(NC(=O)CCN2CC3CN(C(=O)c4cc(Cl)ccc4Cl)CC3C2)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 2/20 0.48
LMNA P02545 3/20 0.47
TP53 P04637 3/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HCRTR1 O43613 1/20 0.45
HCRTR2 O43614 1/20 0.45
UBE2M P61081 1/20 0.44
DCUN1D1 Q96GG9 1/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.43
POLB P06746 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690677 0.92 POLB (0.48) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4692391 0.90 CYP2C9 (0.47) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4692884 0.87 LMNA (0.48) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4695934 0.87 HCRTR1 (0.47) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4694082 0.87 MEN1 (0.47) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4690733 0.86 HCRTR1 (0.46) CYP2C9CYP2C19KMT2ATP53GAA
SCHEMBL4694374 0.86 KMT2A (0.48) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4694967 0.86 KMT2A (0.48) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4692708 0.86 CYP1A2 (0.49) CYP2C9CYP2C19KMT2ALMNATP53
SCHEMBL4691866 0.86 KMT2A (0.47) CYP2C9CYP2C19KMT2ALMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed