SCHEMBL4692391

SCHEMBL4692391

CSc1ccc(Cl)c(C(=O)N2CC3CN(CCC(=O)Nc4ccc(C)c(Cl)c4)CC3C2)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
TP53 P04637 1/20 0.44
MAPT P10636 4/20 0.43
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 2/20 0.43
MAPK1 P28482 2/20 0.43
MEN1 O00255 1/20 0.43
ALOX15 P16050 1/20 0.43
GAA P10253 1/20 0.41
LMNA P02545 4/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 1/20 0.41
GLA P06280 1/20 0.41
HTT P42858 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692691 0.90 CYP2C9 (0.49) CYP2C9CYP2C19TP53MAPTKMT2A
SCHEMBL4691546 0.85 SMN1; SMN2 (0.40) MAPTALDH1A1KMT2AGAALMNA
SCHEMBL4695934 0.85 HCRTR1 (0.47) CYP2C9CYP2C19TP53MAPTALDH1A1
SCHEMBL4692884 0.85 LMNA (0.48) CYP2C9CYP2C19TP53MAPTALDH1A1
SCHEMBL4694082 0.84 MEN1 (0.47) CYP2C9CYP2C19TP53MAPTKMT2A
SCHEMBL4690733 0.84 HCRTR1 (0.46) CYP2C9CYP2C19TP53MAPTKMT2A
SCHEMBL4690677 0.84 POLB (0.48) CYP2C9CYP2C19TP53MAPTKMT2A
SCHEMBL4692701 0.83 CYP2C9 (0.51) CYP2C9CYP2C19TP53MAPTALDH1A1
SCHEMBL4691866 0.83 KMT2A (0.47) CYP2C9CYP2C19TP53MAPTALDH1A1
SCHEMBL4694352 0.83 KMT2A (0.47) CYP2C9CYP2C19TP53ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed