SCHEMBL4692902

SCHEMBL4692902

NC(=O)c1oc(-c2ccccc2)cc1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HCRTR2 O43614 15/20 0.36
HCRTR1 O43613 14/20 0.36
SCD O00767 2/20 0.33
SCD5 Q86SK9 2/20 0.33
SLC9A1 P19634 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694116 0.81 HCRTR2 (0.38) HCRTR2HCRTR1
SCHEMBL4691798 0.80 HCRTR1 (0.42) HCRTR2HCRTR1
SCHEMBL4691643 0.78 LMNA (0.43) KDM4EALDH1A1HCRTR2HCRTR1
SCHEMBL4695411 0.78 CHRNA4 (0.40) ALDH1A1HCRTR2HCRTR1
SCHEMBL4694094 0.78 CHRNB2 (0.44) ALDH1A1
SCHEMBL4691191 0.77 HCRTR1 (0.40) HCRTR2HCRTR1
SCHEMBL4691531 0.77 HCRTR1 (0.41) HCRTR2HCRTR1
SCHEMBL4692504 0.77 HCRTR1 (0.44) KDM4EALDH1A1HCRTR2HCRTR1
SCHEMBL4690347 0.77 HCRTR2 (0.42) HCRTR2HCRTR1
SCHEMBL4693281 0.77 CHRNB2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed