SCHEMBL4693028

SCHEMBL4693028

CC(C)(C)OC(=O)CN(C(=O)C(F)(F)F)c1scc(Br)c1CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSTO1 P78417 1/20 0.36
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4149093 0.88 MEN1 (0.33) GSTO1
SCHEMBL4692615 0.85 HDAC4 (0.32)
SCHEMBL4138268 0.80 MEN1 (0.35) GSTO1
SCHEMBL10866253 0.70 MEN1 (0.47) GSTO1
SCHEMBL4695111 0.69 MTNR1A (0.34) MTNR1AMTNR1B
SCHEMBL4693024 0.65
SCHEMBL3905163 0.65 KMT2A (0.40) GSTO1
SCHEMBL10243532 0.62 CTSK (0.46)
SCHEMBL4697289 0.61 AKR1B1 (0.36)
SCHEMBL4811503 0.60 TSHR (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed