SCHEMBL4693310

SCHEMBL4693310

Cc1ccc(NCCCN2CC3CN(C(=O)c4c(Cl)ccc(C)c4F)CC3C2)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.42
MAPT P10636 4/20 0.40
ALDH1A1 P00352 4/20 0.40
LMNA P02545 2/20 0.40
GAA P10253 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
RAB9A P51151 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
CCL5 P13501 2/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694758 0.93 MAPT (0.40) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4695365 0.89 BRAF (0.39) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4691999 0.89 MAPT (0.51) CCR5MAPTALDH1A1GAAHCRTR1
SCHEMBL4694791 0.89 MAPT (0.47) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4694816 0.89 CCR5 (0.44) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4691511 0.89 CCR5 (0.54) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4694337 0.88 CCR5 (0.43) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4690404 0.88 CCR5 (0.41) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL3281865 0.88 CCR5 (0.52) CCR5MAPTALDH1A1LMNAGAA
SCHEMBL4695514 0.88 MAPT (0.40) CCR5MAPTALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed