SCHEMBL4694337

SCHEMBL4694337

Cc1cc(C)c(C(=O)N2CC3CN(CCCNc4ccc(C)c(Cl)c4)CC3C2)c(C)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.43
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
ALDH1A1 P00352 5/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
AGTR1 P30556 1/20 0.40
HTT P42858 2/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690404 0.94 CCR5 (0.41) CCR5ALDH1A1MAPTLMNAAGTR1
SCHEMBL3281865 0.92 CCR5 (0.52) CCR5HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4692332 0.91 CCR5 (0.51) CCR5HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4692761 0.89 MAPT (0.46) CCR5ALDH1A1MAPTLMNAHTT
SCHEMBL4694791 0.88 MAPT (0.47) CCR5HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4693310 0.88 CCR5 (0.42) CCR5HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4691511 0.88 CCR5 (0.54) CCR5HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4690742 0.88 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1MAPTLMNA
SCHEMBL4694816 0.88 CCR5 (0.44) CCR5HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4690482 0.88 CCR5 (0.43) CCR5HCRTR1HCRTR2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed