SCHEMBL4694077

SCHEMBL4694077

COc1c(Br)cccc1C(=O)N1CC2CN(CCCNC(=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 7/20 0.43
DRD2 P14416 11/20 0.42
DRD4 P21917 11/20 0.42
SIGMAR1 Q99720 2/20 0.42
SLC29A1 Q99808 1/20 0.42
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
SMYD2 Q9NRG4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692997 0.90 SMYD2 (0.41) DRD3DRD2DRD4SMYD2
SCHEMBL4693959 0.90 HCRTR1 (0.45) DRD3DRD2DRD4SIGMAR1SMYD2
SCHEMBL3284096 0.88 SMYD2 (0.44) DRD3DRD2DRD4SMYD2
SCHEMBL4694080 0.87 HCRTR1 (0.40) DRD3DRD2DRD4SIGMAR1
SCHEMBL4691761 0.86 SLC6A2 (0.44) DRD3DRD2DRD4SMYD2
SCHEMBL4691218 0.86 DRD2 (0.45) DRD3DRD2DRD4CYP2D6CYP2C9
SCHEMBL4692672 0.86 SMYD2 (0.45) DRD3DRD2DRD4SMYD2
SCHEMBL4693332 0.85 SLC6A4 (0.45) DRD3DRD2DRD4SIGMAR1SMYD2
SCHEMBL4692216 0.85 SLC6A2 (0.43) DRD3DRD2DRD4SMYD2
SCHEMBL4692347 0.84 DRD2 (0.42) DRD3DRD2DRD4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed