SCHEMBL4692997

SCHEMBL4692997

Cc1ccc(C(=O)NCCCN2CC3CN(C(=O)c4cccc(Br)c4C)CC3C2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 1/20 0.41
SLC6A4 P31645 2/20 0.40
SLC6A2 P23975 1/20 0.40
DRD2 P14416 3/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ADRA1A P35348 1/20 0.40
DRD3 P35462 1/20 0.40
DRD4 P21917 2/20 0.39
MAPK14 Q16539 1/20 0.39
RAD52 P43351 1/20 0.39
CCR5 P51681 1/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GAA P10253 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693959 0.93 HCRTR1 (0.45) SMYD2SLC6A4SLC6A2DRD2LMNA
SCHEMBL4691761 0.93 SLC6A2 (0.44) SMYD2SLC6A4SLC6A2DRD2LMNA
SCHEMBL3284096 0.90 SMYD2 (0.44) SMYD2SLC6A4SLC6A2DRD2LMNA
SCHEMBL4694077 0.90 DRD3 (0.43) SMYD2DRD2DRD3DRD4
SCHEMBL4692672 0.89 SMYD2 (0.45) SMYD2SLC6A4SLC6A2DRD2LMNA
SCHEMBL4696106 0.89 LMNA (0.41) SMYD2LMNASMN1; SMN2MAPK14RAD52
SCHEMBL4693332 0.88 SLC6A4 (0.45) SMYD2SLC6A4SLC6A2DRD2LMNA
SCHEMBL4692216 0.88 SLC6A2 (0.43) SMYD2SLC6A4SLC6A2DRD2LMNA
SCHEMBL4692347 0.87 DRD2 (0.42) SLC6A4SLC6A2DRD2LMNASMN1; SMN2
SCHEMBL4690664 0.87 SMYD2 (0.43) SMYD2SLC6A4SLC6A2DRD2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed