Cyclopentane

Cyclopentane

SCHEMBL4694254

C1CCCC1.O=C(O)NC(CCN1CC2CN(C(=O)c3cccnc3)C[C@@H]2C1)c1ccccc1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.60
CHRNB2 P17787 1/20 0.50
CHRNB4 P30926 1/20 0.50
CHRNA3 P32297 1/20 0.50
CHRNA7 P36544 1/20 0.50
CHRNA4 P43681 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5422985 0.90 CCR5 (0.68) CCR5
Cyclopentane SCHEMBL4696541 0.83 CCR5 (0.69) CCR5
SCHEMBL3283162 0.83 CHRNB2 (0.54) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
Cyclopentane SCHEMBL4695120 0.82 CCR5 (0.63) CCR5
Cyclopentane SCHEMBL4691110 0.82 CCR5 (0.64) CCR5
Cyclopentane SCHEMBL4697136 0.81 CCR5 (0.59) CCR5
SCHEMBL4694961 0.81 CCR5 (0.72) CCR5
SCHEMBL4694960 0.81 CCR5 (0.72) CCR5
Cyclopentane SCHEMBL4694862 0.80 CCR5 (0.65) CCR5
Cyclopentane SCHEMBL4695484 0.80 CCR5 (0.78) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed