SCHEMBL4694527

SCHEMBL4694527

Cc1ccc(NC(=O)CCN2CC3CN(C(=O)c4cc5ccccc5[nH]4)CC3C2)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 6/20 0.53
DRD2 P14416 2/20 0.48
HRH4 Q9H3N8 6/20 0.46
HRH3 Q9Y5N1 1/20 0.46
AKR1C3 P42330 3/20 0.46
MEN1 O00255 1/20 0.43
HCRTR1 O43613 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694532 0.86 DRD3 (0.53) DRD3DRD2HRH4HRH3AKR1C3
SCHEMBL4693095 0.85 TP53 (0.45) MEN1KMT2ALMNA
SCHEMBL4692884 0.83 LMNA (0.48) MEN1KMT2ALMNA
SCHEMBL4693483 0.82 HCRTR1 (0.48) MEN1HCRTR1KMT2ALMNA
SCHEMBL4695277 0.82 MAOB (0.48) DRD3DRD2LMNA
SCHEMBL4692164 0.82 LMNA (0.48) DRD3DRD2MEN1KMT2ALMNA
SCHEMBL3281859 0.82 CCR5 (0.52) MEN1HCRTR1KMT2ALMNA
SCHEMBL4693797 0.81 MAPT (0.51) MEN1KMT2ALMNA
SCHEMBL4695828 0.81 HRH3 (0.46) HRH3MEN1KMT2ALMNA
SCHEMBL4694219 0.80 LMNA (0.46) MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed