SCHEMBL4694846

SCHEMBL4694846

Cc1ccc(NCCCN2CC3CN(C(=O)c4cc5ccccc5nc4C)CC3C2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 5/20 0.40
ALDH1A1 P00352 4/20 0.40
HCRTR1 O43613 4/20 0.39
HCRTR2 O43614 4/20 0.39
POLB P06746 1/20 0.38
CCR5 P51681 2/20 0.38
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SLC6A4 P31645 2/20 0.37
F2 P00734 1/20 0.37
AGTR1 P30556 1/20 0.37
NTRK1 P04629 1/20 0.36
NTRK2 Q16620 1/20 0.36
UBE2M P61081 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693802 0.87 MEN1 (0.46) SMN1; SMN2MAPTALDH1A1MAPK1KMT2A
SCHEMBL4694844 0.86 POLB (0.45) SMN1; SMN2MAPTALDH1A1POLBMAPK1
SCHEMBL4693334 0.86 ALDH1A1 (0.45) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4692889 0.86 MAPT (0.45) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4691905 0.84 HCRTR1 (0.47) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4690668 0.84 ALDH1A1 (0.43) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4690545 0.83 KDM4E (0.41) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4693716 0.83 HCRTR1 (0.52) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4693486 0.83 HCRTR1 (0.48) SMN1; SMN2GAAKDM4EMAPTALDH1A1
SCHEMBL4693961 0.83 HCRTR1 (0.46) SMN1; SMN2GAAKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed