SCHEMBL4695320

SCHEMBL4695320

O=C(NC(CCN1CC2CNC[C@H]2[C@H]1C(=O)c1c(F)cccc1Cl)c1ccccc1)c1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.41
ITGB2 P05107 1/20 0.34
ICAM1 P05362 1/20 0.34
ITGAL P20701 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SLC6A9 P48067 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
DCAF1 Q9Y4B6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696921 0.91 CCR5 (0.47) CCR5SLC6A9
SCHEMBL4696511 0.87 CCR5 (0.40) CCR5ITGB2ICAM1ITGAL
SCHEMBL4696469 0.87 CCR5 (0.41) CCR5KMT2AMEN1SMN1; SMN2
SCHEMBL4694830 0.87 CCR5 (0.41) CCR5
SCHEMBL4694831 0.87 CCR5 (0.41) CCR5
SCHEMBL4695429 0.86 CCR5 (0.46) CCR5SLC6A9
SCHEMBL4690656 0.85 CCR5 (0.43) CCR5KMT2A
SCHEMBL4696815 0.84 CCR5 (0.40) CCR5
SCHEMBL4694955 0.82 CCR5 (0.38) CCR5KMT2AMEN1
SCHEMBL4692299 0.79 CCR5 (0.58) CCR5SLC6A9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed