SCHEMBL4695429

SCHEMBL4695429

Cc1ccnc(C)c1C(=O)NC(CCN1CC2CNC[C@H]2[C@H]1C(=O)c1c(F)cccc1Cl)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 14/20 0.46
ITGB1 P05556 2/20 0.41
ITGA4 P13612 2/20 0.41
SLC6A9 P48067 1/20 0.41
UTS2R Q9UKP6 1/20 0.36
P2RX7 Q99572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696921 0.92 CCR5 (0.47) CCR5ITGB1ITGA4SLC6A9UTS2R
SCHEMBL4695320 0.86 CCR5 (0.41) CCR5SLC6A9
SCHEMBL4696469 0.83 CCR5 (0.41) CCR5UTS2R
SCHEMBL4694831 0.83 CCR5 (0.41) CCR5
SCHEMBL4694830 0.83 CCR5 (0.41) CCR5
SCHEMBL4696511 0.82 CCR5 (0.40) CCR5P2RX7
SCHEMBL4696815 0.82 CCR5 (0.40) CCR5
SCHEMBL4690656 0.80 CCR5 (0.43) CCR5
SCHEMBL4690148 0.79 CCR5 (0.67) CCR5
SCHEMBL4690158 0.79 CCR5 (0.67) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed