SCHEMBL4695580

SCHEMBL4695580

Cc1ccc2c3cccc4c(Br)ccc(c5ccc(C)c1c25)c43

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
CYP1B1 Q16678 3/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 3/20 0.37
CYP2A6 P11509 2/20 0.37
BRD1 O95696 1/20 0.35
TAF1 P21675 1/20 0.35
BRPF1 P55201 1/20 0.35
MAPT P10636 4/20 0.33
TP53 P04637 2/20 0.33
MAPK1 P28482 2/20 0.33
LMNA P02545 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17151500 0.89 ALDH1A1 (0.48) ALDH1A1L3MBTL1CYP1B1CYP3A4HPGD
SCHEMBL6808696 0.85 CYP1A2 (0.48) ALDH1A1L3MBTL1CYP1B1CYP3A4HPGD
SCHEMBL3575204 0.84 CYP1A2 (0.45) ALDH1A1CYP1B1HPGDHSD17B10CYP1A2
SCHEMBL29405395 0.84 CYP1A2 (0.45) ALDH1A1CYP1B1HPGDHSD17B10CYP1A2
SCHEMBL2679177 0.84 CYP1A2 (0.45) ALDH1A1CYP1B1HPGDHSD17B10CYP1A2
SCHEMBL29406732 0.84 CYP1A2 (0.45) ALDH1A1CYP1B1HPGDHSD17B10CYP1A2
SCHEMBL5251847 0.83 ALDH1A1 (0.42) ALDH1A1L3MBTL1CYP1B1CYP3A4HPGD
SCHEMBL14227003 0.80 CYP1A2 (0.36) ALDH1A1L3MBTL1CYP1B1HPGDHSD17B10
SCHEMBL9055556 0.78 ALDH1A1 (0.41) ALDH1A1CYP1B1CYP3A4HPGDTSHR
SCHEMBL2779320 0.76 CYP1A2 (0.42) ALDH1A1L3MBTL1CYP3A4HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874773-A1 HEXARYLENE AND PENTARYLENE TETRACARBOXYLIC ACID DIIMIDES BASF AKTIENGESELLSCHAFT (DE) 2008-01-09 EP claimed
WO-2006111511-A1 HEXARYLENE AND PENTARYLENE TETRACARBOXYLIC ACID DIIMIDES BASF AKTIENGESELLSCHAFT (DE) 2006-10-26 WO claimed
EP-1713777-A1 METHOD FOR PRODUCING TERRYLEN-3,4:11,12-TETRACARBON ACID DI-IMIDS BASF AKTIENGESELLSCHAFT (DE) 2006-10-25 EP claimed
WO-2005070894-A1 METHOD FOR PRODUCING TERRYLEN-3,4:11,12-TETRACARBON ACID DI-IMIDS BASF AKTIENGESELLSCHAFT (DE) 2005-08-04 WO claimed
EP-1542975-A2 9-CYANO-SUBSTITUTED PERYLENE-3,4-DICARBOXYLIC ACID MONOIMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-06-22 EP claimed
WO-2004029028-A2 9-CYANO-SUBSTITUTED PERYLENE-3,4-DICARBOXYLIC ACID MONOIMIDES AS DYESTUFFS BASF AKTIENGESELLSCHAFT (DE) 2004-04-08 WO claimed
EP-1206456-A1 THERMOCHROMIC RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2002-05-22 EP claimed
WO-2001016109-A1 THERMOCHROMIC RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2001-03-08 WO claimed
EP-1542975-A2 9-CYANO-SUBSTITUTED PERYLENE-3,4-DICARBOXYLIC ACID MONOIMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-06-22 EP disclosed
WO-2004029028-A2 9-CYANO-SUBSTITUTED PERYLENE-3,4-DICARBOXYLIC ACID MONOIMIDES AS DYESTUFFS BASF AKTIENGESELLSCHAFT (DE) 2004-04-08 WO disclosed