SCHEMBL4695801

SCHEMBL4695801

N#Cc1ccccc1NC1CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 8/20 0.53
CCNT1 O60563 2/20 0.49
CCNK O75909 2/20 0.49
CCNE1 P24864 2/20 0.49
CDK2 P24941 2/20 0.49
CDK9 P50750 2/20 0.49
CDK12 Q9NYV4 2/20 0.49
PRKCZ Q05513 4/20 0.49
DPP4 P27487 1/20 0.46
PRKD2 Q9BZL6 3/20 0.44
KDM1A O60341 1/20 0.43
MAOB P27338 1/20 0.43
PDPK1 O15530 1/20 0.42
RPS6KB1 P23443 1/20 0.42
HTR6 P50406 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21460264 0.91 IRAK4 (0.45) IRAK4CCNT1CCNKCCNE1CDK2
SCHEMBL2666741 0.82 KDM4E (0.53) KMT2A
SCHEMBL7526224 0.82 KMT2A (0.51) KMT2A
SCHEMBL377808 0.81 CTSL (0.42) IRAK4HTR6KMT2A
SCHEMBL3476117 0.81 KDM4E (0.56) KMT2A
SCHEMBL38662424 0.81 PDPK1 (0.44) IRAK4CCNT1CCNKCCNE1CDK2
Hydrochloric Acid SCHEMBL29882259 0.80 CTSL (0.41) IRAK4KDM1AHTR6KMT2A
SCHEMBL24074639 0.79 KMT2A (0.47) KMT2A
SCHEMBL3727731 0.77 PRKCZ (0.52) CDK2PRKCZPRKD2KDM1AMAOB
SCHEMBL8236935 0.77 KDM4E (0.65) PRKCZPRKD2KDM1AMAOBHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973918-A2 DERIVATIVES OF BETA-AMINO ACID AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS RANBAXY LABORATORIES, LTD. (IN) 2008-10-01 EP disclosed
WO-2007077508-A2 DERIVATIVES OF BETA-AMINO ACID AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2007-07-12 WO disclosed