SCHEMBL4696355

SCHEMBL4696355

O=C1CNC(C(=O)O)c2sccc21

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 2/20 0.32
HTT P42858 1/20 0.32
TSHR P16473 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138455 0.82 KMT2A (0.42) NPSR1
SCHEMBL5251738 0.70 TSHR (0.49) TSHRNPSR1
SCHEMBL4894264 0.69 TSHR (0.51) TSHRNPSR1
SCHEMBL7875920 0.67 EGLN1 (0.35) TSHRNPSR1
SCHEMBL4696279 0.66 AGTR2 (0.35) AGTR2HTT
SCHEMBL23829881 0.62
SCHEMBL11559672 0.61 ACE (0.30)
SCHEMBL8379584 0.61 ACE (0.30)
SCHEMBL28154196 0.61 GRIA2 (0.32)
SCHEMBL9207161 0.60 TSHR (0.53) TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed