SCHEMBL4696456

SCHEMBL4696456

COCCCOCCOC(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.42
CHRM2 P08172 2/20 0.42
CHRM4 P08173 2/20 0.42
CHRM5 P08912 2/20 0.42
CHRM1 P11229 2/20 0.42
CHRM3 P20309 2/20 0.42
LMNA P02545 2/20 0.42
CHRNB2 P17787 2/20 0.42
CHRNA4 P43681 2/20 0.42
HTR1A P08908 1/20 0.42
CYP2C19 P33261 1/20 0.42
CHRNA7 P36544 1/20 0.42
ALOX15 P16050 1/20 0.39
ALDH1A1 P00352 5/20 0.38
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CYP3A4 P08684 2/20 0.35
ABCB11 O95342 1/20 0.35
ADRA2B P18089 1/20 0.35
OPRD1 P41143 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29221545 0.89 TSHR (0.46) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL5531906 0.89 TSHR (0.46) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL631206 0.89 TSHR (0.46) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL30678661 0.89 TSHR (0.46) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL4601154 0.87
SCHEMBL499368 0.82
SCHEMBL24835739 0.82 TSHR (0.50) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL31591142 0.82 TSHR (0.50) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL30552236 0.82 TSHR (0.50) TSHRCHRM2CHRM4CHRM5CHRM1
SCHEMBL11554689 0.81 TSHR (0.48) TSHRCHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987037-A2 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-11-05 EP disclosed
WO-2007097470-A2 FUSED NITROGEN- COMPRISING HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-30 WO disclosed