SCHEMBL469821

SCHEMBL469821

CC(C)(C)OC(=O)N1CCCC1c1cc(F)cc(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 5/20 0.46
GPR119 Q8TDV5 3/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17067861 1.00 RIPK1 (0.46) RIPK1GPR119ALDH1A1LMNANPSR1
SCHEMBL2695225 0.83 RIPK1 (0.50) RIPK1ALDH1A1LMNANPSR1NPC1
SCHEMBL933084 0.83 RIPK1 (0.50) RIPK1ALDH1A1LMNANPSR1NPC1
SCHEMBL455372 0.83 AR (0.39) RIPK1GPR119
SCHEMBL12477574 0.83 AR (0.39) RIPK1GPR119
SCHEMBL456382 0.83 RIPK1 (0.50) RIPK1
SCHEMBL469718 0.83 RIPK1 (0.50) RIPK1
SCHEMBL430865 0.82 AR (0.40) RIPK1GPR119
SCHEMBL457104 0.82 AR (0.40) RIPK1GPR119
SCHEMBL12688003 0.82 AR (0.40) RIPK1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012116217-A1 COMPOUNDS AND COMPOSITIONS AS TRK INHIBITORS IRM LLC (BM) 2012-08-30 WO disclosed
WO-2012034091-A1 IMIDAZO [1, 2] PYRIDAZIN COMPOUNDS AND COMPOSITIONS AS TRK INHIBITORS IRM LLC (BM) 2012-03-15 WO disclosed