SCHEMBL469718

SCHEMBL469718

CC(C)(C)OC(=O)N1CCC[C@@H]1c1cccc(C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.50
SCD O00767 2/20 0.49
SCD5 Q86SK9 2/20 0.49
DRD2 P14416 5/20 0.47
DRD3 P35462 5/20 0.47
ROCK2 O75116 5/20 0.46
HCRTR2 O43614 1/20 0.44
CYP2D6 P10635 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
CASP1 P29466 1/20 0.44
NOTCH1 P46531 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456382 1.00 RIPK1 (0.50) RIPK1SCDSCD5DRD2DRD3
SCHEMBL31421008 0.85 GPR119 (0.51) RIPK1SCD5
SCHEMBL878861 0.83 NPSR1 (0.56) RIPK1SCD5ROCK2TSHR
SCHEMBL469821 0.83 RIPK1 (0.46) RIPK1
SCHEMBL17067861 0.83 RIPK1 (0.46) RIPK1
SCHEMBL17067869 0.82 RIPK1 (0.73) RIPK1SCD5TSHR
SCHEMBL22505052 0.82 USP30 (0.53) RIPK1SCD5ROCK2TSHR
SCHEMBL21198773 0.82 RIPK1 (0.53) RIPK1TSHR
SCHEMBL21207072 0.82 RIPK1 (0.53) RIPK1TSHR
SCHEMBL469686 0.82 RIPK1 (0.73) RIPK1SCD5TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012034095-A1 COMPOUNDS AND COMPOSITIONS AS TRK INHIBITORS IRM LLC (BM) 2012-03-15 WO disclosed