SCHEMBL469851

SCHEMBL469851

O=C(O)NNC(=S)Nc1ccc(F)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 3/20 0.73
GAA P10253 7/20 0.64
PLK4 O00444 1/20 0.61
DAPK3 O43293 1/20 0.61
RPS6KA5 O75582 1/20 0.61
MAP4K4 O95819 1/20 0.61
ERBB2 P04626 1/20 0.61
PRKCG P05129 1/20 0.61
PIM1 P11309 1/20 0.61
PHKG2 P15735 1/20 0.61
CDK2 P24941 1/20 0.61
AXL P30530 1/20 0.61
AKT1 P31749 1/20 0.61
AKT2 P31751 1/20 0.61
PRKCI P41743 1/20 0.61
SYK P43405 1/20 0.61
MAPKAPK2 P49137 1/20 0.61
CLK2 P49760 1/20 0.61
GSK3A P49840 1/20 0.61
GSK3B P49841 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL469849 0.88 NOX1 (0.84) NOX1GAAPLK4DAPK3RPS6KA5
SCHEMBL19277757 0.84 KMT2A (0.74) NOX1GAAPLK4DAPK3RPS6KA5
SCHEMBL28641155 0.84 NOX1 (0.66) NOX1GAAPLK4DAPK3RPS6KA5
SCHEMBL28679366 0.81 GAA (0.71) NOX1GAAPLK4DAPK3RPS6KA5
SCHEMBL10099725 0.80 GAA (0.83) NOX1GAAMEN1KMT2APOLB
SCHEMBL935849 0.78 ALDH1A1 (0.64) GAAMEN1KMT2APOLBRAB9A
SCHEMBL18031169 0.76 GAA (1.00) NOX1GAAMEN1KMT2APOLB
SCHEMBL10710275 0.76 NOX1 (0.85) NOX1GAAMEN1KMT2APOLB
SCHEMBL8014406 0.76 GAA (0.81) NOX1GAAMEN1KMT2ARAB9A
SCHEMBL457622 0.76 GAA (0.64) NOX1GAAPLK4DAPK3RPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033601-A1 THIOSEMICARBAZONES WITH MDR1 - INVERSE ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2012-03-15 WO disclosed