SCHEMBL469867

SCHEMBL469867

COC(=O)c1cc2c(cc1F)CCC(NS(=O)(=O)c1ccc(C)cc1)C2

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 7/20 0.63
ALDH1A1 P00352 4/20 0.47
TSHR P16473 3/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.44
HDAC6 Q9UBN7 1/20 0.43
HPGD P15428 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL464353 0.91 HDAC8 (0.76) HDAC8ALDH1A1TSHRMAPTHDAC6
SCHEMBL469843 0.81 HDAC8 (0.47) HDAC8ALDH1A1TSHRHDAC6HPGD
SCHEMBL415810 0.80 HDAC8 (0.48) HDAC8ALDH1A1TSHRHDAC6HPGD
SCHEMBL446824 0.77 HDAC8 (1.00) HDAC8MAPTHDAC6POLB
SCHEMBL21292761 0.76 KMT2A (0.62) ALDH1A1TSHRMAPTHPGDKMT2A
SCHEMBL10463170 0.75 POLB (0.50) HDAC8ALDH1A1TSHRCYP3A4HPGD
SCHEMBL8384541 0.73 PSEN1 (0.64) HDAC8ALDH1A1TSHRCYP3A4KMT2A
SCHEMBL415355 0.73 MTNR1A (0.41) HDAC8GAA
SCHEMBL416742 0.72 MAPT (0.47) ALDH1A1MAPTHSD17B10
SCHEMBL355191 0.72 HDAC8 (0.59) HDAC8ALDH1A1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031993-A1 NOVEL N-HYDROXY-BENZAMIDES FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2012-03-15 WO disclosed