SCHEMBL469843

SCHEMBL469843

CNC1CCc2cc(F)c(C(=O)OC)cc2C1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 4/20 0.47
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
MTNR1A P48039 3/20 0.40
MTNR1B P49286 3/20 0.40
CA1 P00915 6/20 0.38
CA2 P00918 6/20 0.38
ACHE P22303 6/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HDAC6 Q9UBN7 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415810 0.88 HDAC8 (0.48) HDAC8MTNR1AMTNR1BCA1CA2
SCHEMBL415355 0.83 MTNR1A (0.41) HDAC8DRD2MTNR1AMTNR1BCA1
SCHEMBL416742 0.82 MAPT (0.47) DRD2DRD3ACHEALDH1A1HSD17B10
SCHEMBL469741 0.82 HDAC8 (0.53) HDAC8HDAC6
SCHEMBL469867 0.81 HDAC8 (0.63) HDAC8ALDH1A1HPGDTSHRHSD17B10
SCHEMBL464353 0.80 HDAC8 (0.76) HDAC8ALDH1A1HPGDTSHRHSD17B10
SCHEMBL883735 0.78 RAB9A (0.42) CA1CA2ALDH1A1HPGDTSHR
SCHEMBL469781 0.75 MTNR1A (0.51) HDAC8DRD2DRD4DRD3MTNR1A
SCHEMBL17269807 0.74 ALDH1A1 (0.42) DRD2DRD4DRD3MTNR1AMTNR1B
SCHEMBL803162 0.73 ACHE (0.42) ACHEALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031993-A1 NOVEL N-HYDROXY-BENZAMIDES FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2012-03-15 WO disclosed