SCHEMBL4700092

SCHEMBL4700092

COC(=O)c1ccc(-c2cccc(O)c2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.65
HSD17B1 P14061 5/20 0.59
HSD17B2 P37059 5/20 0.59
CYP3A4 P08684 2/20 0.59
CYP2C9 P11712 1/20 0.59
CA12 O43570 3/20 0.58
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
CA9 Q16790 3/20 0.58
CA14 Q9ULX7 2/20 0.58
CA7 P43166 1/20 0.58
ERN1 O75460 2/20 0.56
HPGDS O60760 2/20 0.52
PLAU P00749 2/20 0.52
TSHR P16473 1/20 0.50
PTPN1 P18031 1/20 0.50
CYP17A1 P05093 1/20 0.49
CYP19A1 P11511 1/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31337006 1.00 EGFR (0.65) EGFRHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL28189889 0.89 EGFR (0.68) EGFRCA12CA1CA2CA9
SCHEMBL6434807 0.88 ERN1 (0.61) HSD17B1HSD17B2CYP3A4CYP2C9CA12
SCHEMBL27589486 0.87 TSHR (0.64) EGFRCA12CA1CA2CA9
SCHEMBL68931 0.86 CA12 (0.69) EGFRCA12CA1CA2CA9
SCHEMBL6138470 0.83 EGFR (0.60) EGFRHSD17B1HSD17B2CA12CA1
SCHEMBL1661764 0.83 CA12 (0.66) EGFRCA12CA1CA2CA9
SCHEMBL30443216 0.83 CA12 (0.66) EGFRCA12CA1CA2CA9
SCHEMBL31298127 0.83 EGFR (0.60) EGFRHSD17B1HSD17B2CA12CA1
SCHEMBL21228271 0.82 CA12 (0.54) EGFRHSD17B1HSD17B2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506195-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2008-10-29 EP disclosed
US-20060058553-A1 Novel bicyclic hydroxamates as inhibitors of histone deacetylase AXYS PHARMACEUTICALS, INC. (US) 2006-03-16 US disclosed
EP-1506195-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2005-02-16 EP disclosed
EP-1472216-A2 NOVEL BICYCLIC HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE Axys Pharmaceuticals (US) 2004-11-03 EP disclosed
US-6806265-B2 FOR THERAPY AND PROPHYLAXIS OF HIV INFECTION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-10-19 US disclosed
US-20040006071-A1 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2004-01-08 US disclosed
WO-2003097644-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2003-11-27 WO disclosed
WO-2003066579-A2 NOVEL BICYCLIC HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE AXYS PHARMACEUTICALS (US) 2003-08-14 WO disclosed
US-5298593-A Polymerization of ester monomer, aromatic dicarboxylic acid, and oxyaromatic carboxylic acid MITSUBISHI PETROCHEMICAL COMPANY, LTD. (JP) 1994-03-29 US disclosed
EP-0520428-A2 Method of producing thermotropic liquid crystalline polyester MITSUBISHI CHEMICAL CORPORATION (JP) 1992-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040006071-A1 Non-nucleoside reverse transcriptase inhibitors CBR1, POLR2H, SUB1 EGFR 2236/4885HSD17B1 75/4885HSD17B2 194/4885
US-20060058553-A1 Novel bicyclic hydroxamates as inhibitors of histone deacetylase HDAC1, HDAC2, HDAC11 EGFR 4392/4885HSD17B1 522/4885HSD17B2 715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.