SCHEMBL21228271

SCHEMBL21228271

CC(C)(C)OC(=O)c1ccc(-c2cccc(O)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
HSD17B1 P14061 8/20 0.53
HSD17B2 P37059 8/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2C9 P11712 1/20 0.53
HPGDS O60760 2/20 0.46
CYP17A1 P05093 2/20 0.46
EGFR P00533 2/20 0.46
CYP19A1 P11511 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2076830 0.88 CA12 (0.65) CA12CA1CA2CA9CA14
SCHEMBL19497926 0.83 CA12 (0.63) CA12CA1CA2CA9CA14
SCHEMBL6355405 0.83 CA12 (0.63) CA12CA1CA2CA9CA14
SCHEMBL28943519 0.83 CA12 (0.52) CA12CA1CA2CA9CA14
SCHEMBL6350965 0.83 CA12 (0.71) CA12CA1CA2CA9CA14
SCHEMBL31337006 0.82 EGFR (0.65) CA12CA1CA2CA9CA14
SCHEMBL4700092 0.82 EGFR (0.65) CA12CA1CA2CA9CA14
SCHEMBL2344130 0.82 SLC7A5 (0.52) CA12CA1CA2CA9CA14
SCHEMBL68806 0.82 ESR1 (0.53) CA12CA1CA2CA9CYP3A4
SCHEMBL18608496 0.81 RXRA (0.53) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019149205-A1 BENZOHETEROARYL DERIVATIVE AND PREPARATION METHOD AND MEDICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2019-08-08 WO disclosed