SCHEMBL4700523

SCHEMBL4700523

C=CCc1ccc(Br)s1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6292229 0.83 ALDH1A1 (0.34)
SCHEMBL28887753 0.74 KDM4E (0.41)
SCHEMBL28820704 0.73
SCHEMBL7087320 0.73
SCHEMBL974768 0.73
SCHEMBL18770037 0.72 CES2 (0.38)
SCHEMBL13049960 0.72 KDM4E (0.45)
SCHEMBL1414863 0.72 KDM4E (0.45)
SCHEMBL627336 0.71 ALDH1A1 (0.33)
SCHEMBL13873989 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654298-B1 PROCESS OF PREPARING REGIOREGULAR POLYMERS MERCK PATENT GMBH (DE) 2008-10-01 EP disclosed
US-20080164465-A1 Electronic Device KONINKLIJKE PHILIPS ELECTRONICS, N.V. (NL) 2008-07-10 US disclosed
EP-1854159-A1 ELECTRONIC DEVICE Koninklijke Philips Electronics N.V. (NL) 2007-11-14 EP disclosed
US-7294288-B2 Process of preparing regioregular polymers MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2007-11-13 US disclosed
WO-2006087680-A1 ELECTRONIC DEVICE KONINKLIJKE PHILIPS ELECTRONICS N.V. (NL) 2006-08-24 WO disclosed
EP-1654298-A2 PROCESS OF PREPARING REGIOREGULAR POLYMERS MERCK PATENT GmbH (DE) 2006-05-10 EP disclosed
US-20050080219-A1 Process of preparing regioregular polymers MERCK PATENT GMBH (DE) 2005-04-14 US disclosed
WO-2005014691-A2 PROCESS OF PREPARING REGIOREGULAR POLYMERS MERCK PATENT GMBH (DE) 2005-02-17 WO disclosed
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed