SCHEMBL470067

SCHEMBL470067

Cc1cc(-c2cnc3c(NCCN4CCOCC4)cc(Oc4ccc(F)c(F)c4)nn23)ccc1C(N)=O

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TTK P33981 17/20 0.55
CYP3A4 P08684 1/20 0.45
FYN P06241 1/20 0.44
SCN9A Q15858 1/20 0.42
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17425425 0.92 TTK (0.58) TTKCYP3A4FYN
SCHEMBL10279721 0.91 TTK (0.57) TTKCYP3A4FYN
SCHEMBL17590099 0.91 TTK (0.53) TTKCYP3A4SCN9ACSF1R
SCHEMBL17590100 0.91 TTK (0.58) TTKCYP3A4FYNSCN9ACSF1R
SCHEMBL17416389 0.91 TTK (0.68) TTKCYP3A4
SCHEMBL470204 0.88 TTK (0.55) TTKCYP3A4FYNSCN9ACSF1R
SCHEMBL470206 0.87 TTK (0.65) TTK
SCHEMBL470099 0.86 TTK (0.53) TTKCYP3A4FYNCSF1R
SCHEMBL17590107 0.86 TTK (0.58) TTKFYN
SCHEMBL10279537 0.86 TTK (0.60) TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9255100-B2 Substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-02-09 US disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed