SCHEMBL470229

SCHEMBL470229

Cc1cc(C)c(N2CCN(C(=O)OC(C)(C)C)CC2)cc1NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
BACE1 P56817 4/20 0.45
LMNA P02545 4/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 1/20 0.43
NAMPT P43490 1/20 0.42
GPR119 Q8TDV5 1/20 0.42
F13A1 P00488 1/20 0.41
TGM2 P21980 1/20 0.41
TGM1 P22735 1/20 0.41
CYP2C19 P33261 2/20 0.41
SMARCA2 P51531 1/20 0.41
SMARCA4 P51532 1/20 0.41
PBRM1 Q86U86 1/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29796094 0.89 BACE1 (0.48) MEN1KMT2ABACE1LMNANPSR1
SCHEMBL470212 0.89 MEN1 (0.51) MEN1KMT2ABACE1LMNANPSR1
SCHEMBL470218 0.89 BACE1 (0.48) MEN1KMT2ABACE1LMNANPSR1
SCHEMBL457432 0.89 MEN1 (0.51) MEN1KMT2ABACE1LMNANPSR1
SCHEMBL2365831 0.84 LMNA (0.50) MEN1KMT2ALMNAMAPTSMN1; SMN2
SCHEMBL457220 0.83 MAPT (0.52) MEN1KMT2ALMNANPSR1MAPT
SCHEMBL470197 0.81 MEN1 (0.47) MEN1KMT2ABACE1LMNANPSR1
SCHEMBL31129872 0.79 SMARCA2 (0.52) MEN1KMT2ABACE1LMNAMAPT
SCHEMBL463132 0.79 BACE1 (0.49) MEN1KMT2ABACE1LMNANPSR1
SCHEMBL470227 0.79 BACE1 (0.47) MEN1KMT2ABACE1LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed