SCHEMBL4702575

SCHEMBL4702575

CCOc1cc(CN(c2nccc(O)n2)C2CCNCC2)cc(OCC)c1N

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 9/20 0.45
SLC6A4 P31645 9/20 0.45
SLC6A3 Q01959 9/20 0.45
IKBKB O14920 8/20 0.39
KCNH2 Q12809 1/20 0.34
SSTR5 P35346 1/20 0.33
CRHR1 P34998 1/20 0.32
TACR1 P25103 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4702470 0.86 SLC6A4 (0.48) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4705296 0.85 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4703738 0.78 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3
SCHEMBL4704998 0.77 KDM4E (0.37) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4704686 0.75 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4705309 0.75 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3KCNH2SSTR5
SCHEMBL4705827 0.75 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3KCNH2SSTR5
SCHEMBL3971524 0.75 MAPK1 (0.36) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL3973888 0.74 IKBKB (0.40) SLC6A2SLC6A4SLC6A3IKBKB
SCHEMBL4001474 0.73 HTR1F (0.37) SLC6A2SLC6A4SLC6A3IKBKBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed