SCHEMBL4704686

SCHEMBL4704686

CCOc1cc(CN(c2nccc(N)n2)C2CCNCC2)ccc1OC(CC)CC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.45
SLC6A4 P31645 11/20 0.45
SLC6A3 Q01959 9/20 0.45
ADRA2A P08913 2/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
IKBKB O14920 1/20 0.35
MCHR1 Q99705 1/20 0.34
KCNH2 Q12809 2/20 0.33
CYP3A4 P08684 2/20 0.32
MAPK1 P28482 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
DRD1 P21728 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4702575 0.75 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4702470 0.74 SLC6A4 (0.48) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4705848 0.73 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKBREN
SCHEMBL4701133 0.70 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3IKBKBTSHR
SCHEMBL4701120 0.70 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3KCNH2SMN1; SMN2
SCHEMBL4705296 0.70 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4706328 0.70 SLC6A4 (0.44) SLC6A2SLC6A4SLC6A3KCNH2SMN1; SMN2
SCHEMBL4701500 0.69 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKB
SCHEMBL3939023 0.69 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL4704338 0.69 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed