SCHEMBL4704596

SCHEMBL4704596

CN1CCN(c2nc(-c3ccc(OC4CCCCC4)cc3)cs2)CC1.N#CCNC(=O)O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSB P07858 15/20 0.57
CTSS P25774 15/20 0.57
CTSL P07711 13/20 0.57
CTSK P43235 5/20 0.57
SMN1; SMN2 Q16637 2/20 0.45
RAB9A P51151 1/20 0.45
KCNH2 Q12809 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703896 0.79 CTSB (0.70) CTSBCTSSCTSLCTSKSMN1; SMN2
SCHEMBL6183485 0.73 CTSB (1.00) CTSBCTSSCTSLCTSK
SCHEMBL4703916 0.73 CTSB (0.54) CTSBCTSSCTSLCTSKKCNH2
SCHEMBL6182464 0.71 CTSK (0.64) CTSBCTSSCTSLCTSK
SCHEMBL7042069 0.71 CTSB (0.51) CTSBCTSSCTSLCTSKSMN1; SMN2
Trifluoroacetic Acid SCHEMBL6182305 0.70 CTSB (0.89) CTSBCTSSCTSLCTSK
SCHEMBL15741078 0.70 SMN1; SMN2 (0.57) SMN1; SMN2RAB9AALDH1A1MAPK1
SCHEMBL15741082 0.70 SMN1; SMN2 (0.57) SMN1; SMN2RAB9AALDH1A1MAPK1
SCHEMBL4698741 0.70 CTSB (0.58) CTSBCTSSCTSLCTSKSMN1; SMN2
SCHEMBL1841459 0.70 CTSK (0.53) CTSBCTSSCTSLCTSKSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP claimed