SCHEMBL4705486

SCHEMBL4705486

O=C(O)N(CCc1ccc(Cl)c(CO)c1)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 4/20 0.41
REN P00797 11/20 0.39
KCNH2 Q12809 3/20 0.38
MBTPS1 Q14703 2/20 0.38
CYP3A4 P08684 3/20 0.38
OPRM1 P35372 1/20 0.37
SMYD2 Q9NRG4 1/20 0.36
TACR1 P25103 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682630 0.83 REN (0.46) RENKCNH2CYP3A4TACR1
SCHEMBL1750990 0.82 REN (0.39) C5AR1RENKCNH2CYP3A4
SCHEMBL4704492 0.81 SMYD2 (0.39) C5AR1KCNH2MBTPS1CYP3A4OPRM1
SCHEMBL661970 0.78 REN (0.56) RENKCNH2CYP3A4
SCHEMBL18567998 0.76 MBTPS1 (0.51) C5AR1MBTPS1OPRM1TACR1
SCHEMBL4701505 0.76 SIGMAR1 (0.40) OPRM1
SCHEMBL662616 0.73 PSMB5 (0.39) RENKCNH2CYP3A4TACR1
SCHEMBL1750638 0.72 FFAR1 (0.51)
SCHEMBL4682925 0.72 REN (0.56) RENKCNH2CYP3A4
SCHEMBL1751560 0.72 REN (0.40) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893578-A2 NOVEL PIPERIDINE CARBOXYLIC ACID AMIDE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2008-03-05 EP disclosed
WO-2006129237-A2 NOVEL PIPERIDINE CARBOXYLIC ACID AMIDE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2006-12-07 WO disclosed