SCHEMBL470650

SCHEMBL470650

C[C@@H](OS(C)(=O)=O)C1CCN(c2nc(C(C)(C)C)no2)CC1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 14/20 0.39
ALOX5AP P20292 5/20 0.37
GPR183 P32249 1/20 0.34
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470649 0.89 GPR119 (0.40) GPR119ALOX5APGPR183
SCHEMBL384915 0.82 GPR119 (0.59) GPR119GPR183
SCHEMBL386891 0.82 GPR119 (0.59) GPR119GPR183
SCHEMBL470521 0.81 GPR119 (0.39) GPR119GPR183LMNAMAPT
SCHEMBL470684 0.79 GPR119 (0.47) GPR119ALOX5APLMNAMAPT
SCHEMBL2394364 0.75 GPR119 (0.42) GPR119ALOX5APGPR183LMNA
SCHEMBL2371302 0.74 GPR119 (0.49) GPR119GPR183
SCHEMBL12064986 0.74 ALOX5AP (0.40) GPR119ALOX5APGPR183
SCHEMBL356316 0.73 GPR119 (0.59) GPR119ALOX5AP
SCHEMBL19450516 0.72 GPR119 (0.40) GPR119ALOX5APLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147951-A1 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS PROSIDION LIMITED (GB) 2011-12-01 WO disclosed