SCHEMBL4706536

SCHEMBL4706536

CC(C)(C)OC(=O)NCCNCc1cccc(Cl)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.51
DRD2 P14416 2/20 0.50
LMNA P02545 2/20 0.46
MEN1 O00255 1/20 0.46
TSHR P16473 1/20 0.46
KMT2A Q03164 1/20 0.46
NQO2 P16083 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
REN P00797 1/20 0.45
HPGD P15428 1/20 0.44
CYP1A2 P05177 1/20 0.44
GLA P06280 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
IDO1 P14902 2/20 0.43
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5766456 0.91 LMNA (0.54) GAADRD2LMNAMEN1TSHR
SCHEMBL30606607 0.88 LMNA (0.44) GAADRD2LMNAMEN1TSHR
SCHEMBL26599167 0.88 LMNA (0.44) GAADRD2LMNAMEN1TSHR
SCHEMBL29168148 0.85 NQO2 (0.57) GAADRD2LMNAMEN1TSHR
SCHEMBL4708016 0.83 MEN1 (0.52) GAADRD2LMNAMEN1TSHR
SCHEMBL13387818 0.81 MALT1 (0.45) DRD2LMNAMEN1TSHRKMT2A
SCHEMBL5769723 0.81 LMNA (0.54) GAADRD2LMNAMEN1TSHR
SCHEMBL4707006 0.80 CHRM2 (0.49) GAALMNAKMT2ANQO2HPGD
SCHEMBL29761164 0.80 CA12 (0.58) TSHRNQO2CYP2D6MALT1BCHE
SCHEMBL15586460 0.80 NQO2 (0.57) MEN1KMT2ANQO2HPGDATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed