SCHEMBL4706833

SCHEMBL4706833

O=C(c1[nH]c2ccccc2c1CN1CCC(c2c(F)cccc2Cl)CC1)N1CCOCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.46
HTT P42858 2/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP2A13 Q16696 1/20 0.43
KDM4E B2RXH2 2/20 0.42
KMT2A Q03164 3/20 0.41
TSHR P16473 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 4/20 0.40
LMNA P02545 2/20 0.40
USP2 O75604 1/20 0.40
PKM P14618 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
HTR2A P28223 1/20 0.39
MAPT P10636 2/20 0.39
ALOX15 P16050 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707294 0.94 HTT (0.43) MCL1HTTHSD17B10CYP2A13KDM4E
Hydrochloric Acid SCHEMBL4516276 0.93 MCL1 (0.49) MCL1HTTHSD17B10CYP2A13KDM4E
SCHEMBL4778114 0.88 KDM4E (0.42) MCL1HTTKDM4EKMT2ATSHR
SCHEMBL4778117 0.88 KDM4E (0.42) MCL1HTTKDM4EKMT2ATSHR
SCHEMBL4708847 0.87 HTT (0.46) MCL1HTTHSD17B10KMT2ATSHR
Hydrochloric Acid SCHEMBL4527694 0.86 MCL1 (0.58) MCL1HTTHSD17B10KDM4ETSHR
SCHEMBL4706258 0.86 ALDH1A1 (0.47) MCL1HTTHSD17B10KDM4EKMT2A
Hydrochloric Acid SCHEMBL4774402 0.86 ALDH1A1 (0.46) MCL1HTTHSD17B10KDM4EKMT2A
SCHEMBL4514605 0.85 MCL1 (0.51) MCL1HTTHSD17B10KDM4EKMT2A
SCHEMBL4529569 0.85 HTR2A (0.43) MCL1HTTKDM4EKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO claimed
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO disclosed
EP-1873150-A1 Fluorinated indoleamides useful as ligands of the ORL-1 receptor NIKEM RESEARCH S.R.L. (IT) 2008-01-02 EP disclosed