SCHEMBL4707135

SCHEMBL4707135

Cc1ccccc1CN1CCN=C1c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.39
TDO2 P48775 1/20 0.39
CDC7 O00311 5/20 0.37
MAP4K4 O95819 4/20 0.37
PIM1 P11309 4/20 0.37
PRKACA P17612 4/20 0.37
CDK2 P24941 4/20 0.37
GSK3B P49841 4/20 0.37
HIPK2 Q9H2X6 4/20 0.37
CLK4 Q9HAZ1 3/20 0.37
MKNK2 Q9HBH9 3/20 0.37
TACR1 P25103 2/20 0.36
POLB P06746 1/20 0.35
DAPK3 O43293 2/20 0.35
ROCK2 O75116 2/20 0.35
PRKD3 O94806 2/20 0.35
FLT3 P36888 2/20 0.35
CLK2 P49760 2/20 0.35
PRKX P51817 2/20 0.35
JAK3 P52333 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708192 0.89 SMN1; SMN2 (0.40) IDO1TDO2CDC7MAP4K4PIM1
SCHEMBL4707185 0.87 CDC7 (0.37) IDO1TDO2CDC7MAP4K4PIM1
SCHEMBL4707796 0.84 CDC7 (0.39) IDO1TDO2CDC7MAP4K4PIM1
SCHEMBL4707422 0.83 SMN1; SMN2 (0.40) IDO1CDC7MAP4K4PIM1PRKACA
SCHEMBL4705897 0.81 PTAFR (0.40) IDO1CDC7MAP4K4PIM1PRKACA
SCHEMBL4705520 0.81 PTAFR (0.39) IDO1TDO2CDC7MAP4K4PIM1
SCHEMBL4706961 0.80 IDO1 (0.40) IDO1TDO2CDC7MAP4K4PIM1
SCHEMBL4790291 0.80 PTGER4 (0.40) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4705280 0.80 PTGER4 (0.40) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4706420 0.76 IDO1 (0.44) IDO1TDO2CDC7MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed